The Ugly Duckling Metamorphosis: The Ammonia/Formaldehyde Couple Made Possible in Ugi Reactions

Rosalba, T.P.F.; Kas, S.S.A.; Sampaio, A.B.S.; Salvador, C.E.M.; Andrade, C.K.Z. EurJOC 2021, 20, 2831-2842

 

 

 

Phytotoxicity Study of Ortho-Disubstituted Disulfides and Their Acyl Derivatives

Oliveira, S.C.C.; Andrade, C.K.Z.; Varela, R.M.; Molinillo, J.M.G.; Macías, F.A. ACS Omega 2019, 4, 2362-2368

 

 

Structure-activity relationship study of antitrypanosomal chalcone derivatives using multivariate analysis

Gomes, K.S.; Silva, T.A.C.; Oliveira, I.H.; Aguilar, A.M.; Silva, D.O.; Uemi, M.; Silva, W.A.; Melo, L.R.; Andrade, C.K.Z.; Tempone, A.G.; Baldim, J.L.; Lago, J.H.G. Bioorg Med Chem Lett 2019, 29, 1459-1462

 

 

Synthesis of (macro)heterocycles by consecutive/repetitive isocyanide-based multicomponent reactions

Barreto, A.F.S.; Andrade, C.K.Z. Beilstein J Org Chem 2019, 15, 906-930

 

 

A Mild, Fast, and Scalable Synthesis of Substituted α-Acyloxy Ketones via Multicomponent Reaction Using a Continuous Flow Approach

Salvador, C.E.M.; Andrade, C.K.Z. Frontiers in Chem 2019, 7, 531

 

 

Thermostability and physicochemical properties of two macauba oils and their derivatives related to their use as a lubricant base

Matos, P.R.R.; Andrade, C.K.Z.; Rodrigues, J.D.O.; Sales, M.J.A. Almeida, A.S.; Politi, J.R.S. J Therm Anal Calorim 2018, 132, 293-303

 

 

Inhibition of IL-2 Production by Novel Small Molecules using Building Blocks from Reduced Chalcones and a Substituted Proline

Lara, E.F.D.; Silva, W.A.; Guzman, L.; Castro, R.; Andrade, C.K.Z. Santos, L.S. Curr Drug Ther 2018, 13, 130-139

 

 

Microwave-mediated synthesis of a cyclic heptapeptoid through consecutive Ugi reactions

Barreto, A.F.S.; Andrade, C.K.Z. Tetrahedron 2018, 74, 6861-6865

 

 

Microwave-Assisted Aminolysis of Lactones Under Solvent- and Catalyst- Free Conditions

Barreto, A.F.S.; Salvador, C.E.M.; Rosalba, T.P.F.; Andrade, C.K.Z. Current Microwave Chem 2017, 4, 168-172

 

 

Synthesis, Characterization and in vitro Anticancer Activity of Novel 8,4'-Oxyneolignan Analogues

Souza, G.C.; Franchi, G.C.; Nowill, A.E.; Santos, L.S.; Alves, C.N.; Barata, L.E.S.; Andrade, C.K.Z. J Braz Chem Soc 2017, 28, 2229-2243

 

 

Consecutive hydrazino-Ugi-azide reactions: synthesis of acylhydrazines bearing 1,5-disubstituted tetrazoles

Barreto, A.F.S.; Santos, V.A.; Andrade, C.K.Z.  Beilstein J Org Chem 2017, 13, 2596-2602

 

 

Enantioselective Total Syntheses of (R)‐ and (S)‐Naphthotectone, and Stereochemical Assignment of the Natural Product

Vásquez, G.A.G.; Galarza, F.A.D.; Molinillo, J.M.G.; Andrade, C.K.Z.; Macías, F.A. Eur J Org Chem 2016, 2016, 1599-1605

 

 

Applying green processes and techniques to simplify reaction work-ups

Andrade, C.K.Z.; Dar, A.R. Tetrahedron 2016, 72, 7375-7391

 

 

Synthesis of acylhydrazino-peptomers, a new class of peptidomimetics, by consecutive Ugi and hydrazino-Ugi reactions

Barreto, A.F.S.; Santos, V.A.; Andrade, C.K.Z. Beilstein J Org Chem 2016, 12, 2865-2872

In vitro Anti-HMPV Activity of New Synthetic Phenytoin Derivatives

Mendes, G.; Aspesi, G.H.; Arruda, A.L.A.; Romanos, M.T.V.; Andrade, C.K.Z. J Braz Chem Soc 2016, 27, 2-9

A Sequential Ugi Multicomponent/Cu-Catalyzed Azide–Alkyne Cycloaddition Approach for the Continuous Flow Generation of Cyclic Peptoids

Salvador, C.E.M.; Pieber, B.; Neu, P.M.; Torvisco, A., Andrade, C.K.Z; Kappe, C.O. J Org Chem 2015, 80, 4590–4602 

Recent Advances in Using Niobium Compounds as Catalysts in Organic Chemistry

Arpini, B.H.; Bartolomeu, A.A.; Andrade, C.K.Z.; Filho, L.C.S.; Lacerda, V. Curr Org Synt 2015, 12, 570-583

Consecutive isocyanide-based multicomponent reactions: synthesis of cyclic pentadepsipeptoids

Barreto, A.F.S.; Vercillo, O.E.; Wessjohann, L.A.; Andrade, C.K.Z. Beilstein J Org Chem 2014, 10, 1017-1022

Biological and structure-activity evaluation of chalcone derivatives against bacteria and fungi

Silva, W.A.; Andrade, C.K.Z.; Napolitano, H.B.; Vencato, I.; Lariucci, C.; Castro, M.R.C.; Camargo, A.J. J Braz Chem Soc 2013, 24, 133-144

Zingiberenol, (1S,4R,1′S)-4-(1′,5′-Dimethylhex-4′-enyl)-1-methylcyclohex-2-en-1-ol, Identified as the Sex Pheromone Produced by Males of the Rice Stink Bug Oebalus poecilus (Heteroptera: Pentatomidae)

Oliveira, M.W.M.; Borges, M.; Andrade, C.K.Z.; Laumann, R.A.; Barrigossi, J.A.F.; Moraes, M.C.B. J Agric Food Chem 2013, 61, 7777-7785

Practical First Total Synthesis of the Potent Phytotoxic (±)‐Naphthotectone, Isolated from Tectona grandis

Vásquez, G.A.G.; Andrade, C.K.Z.; Molinillo, J.M.G.; Macías, F.A. Eur J Org Chem 2013, 2013, 6175-6180

Evaluation of Spectroscopic and Morphological Properties of PMMA Modified with ILs

Oliveira, V.B.; Pereira, N.S.; Andrade, C.K.Z.; Sales, M.J.A. Macromol Symp 2012, 319, 203-209

Microwave-Assisted Passerini Reactions under Solvent-Free Conditions

Barreto, A.F.S.; Vercillo, O.E.; Andrade, C.K.Z. J Braz Chem Soc 2011, 22, 462-467

Bijvoet in Solution Reveals Unexpected Stereoselectivity in a Michael Addition

Sun, H.; Auvergne, E.J.; Reinscheid, U.M.; Dias, L.C.; Andrade, C.K.Z.; Rocha, R.O.; Griesinger, C. Chem Eur J 2011, 17, 1811-1817

Synthesis and evaluation of quinonoid compounds against tumor cell lines

Silva, E.N.; Cavalcanti, B.C.; Guimarães, T.T.; Pinto, M.C.F.R.; Cabral, I.O.; Pessoa, C.; Lotufo, L.V.C.; Moraes, M.O.; Andrade, C.K.Z.; Santos, M.R.; Simone, C.A.; Goulart, M.O.F.; Pinto, A.V. Eur J Med Chem 2011, 46, 399-410

14th Brazilian Meting on Organic Synthesis: Importância Histórica, Retrospectiva e Perspectivas

Andrade, C.K.Z.; Silva, W.A.; Bakuzis, P. Revista Processos Químicos 2011, 5, 9-22

Inibidores da Proteína Auxiliar Nef do Vírus HIV-1: um Novo Alvo Terapêutico no Tratamento da SIDA

Salvador, C.E.M.; Corrêa, L.Z.A.; Andrade, C.K.Z. Revista Processos Químicos 2011, 5, 56-63

Fast and efficient microwave-assisted synthesis of functionalized peptoids via Ugi reactions

Barreto, A.F.S.; Vercillo, O.E.; Birkett, M.A.; Caulfield, J.C.; Wessjohann, L.A.; Andrade, C.K.Z. Org Biomol Chem 2011, 9, 5024-5027

Thermal study and evaluation of new menthol-based ionic liquids as polymeric additives

Andrade, C.K.Z.; Matos, R.A.F.; Oliveira, V.B.; Durães, J.A.; Sales, M.J.A. J Therm Anal Calorim 2010, 99, 539-543

The evaluation of quinonoid compounds against Trypanosoma cruzi: Synthesis of imidazolic anthraquinones, nor-β-lapachone derivatives and β-lapachone-based 1,2,3-triazoles

Júnior, E.N.S.; Guimarães, T.T.; Barreto, R.F.S.M.; Pinto, M.C.F.R.; Simone, C.A.; Pessoa, C.; Cavalcanti, B.C.; Sabino, J.R.; Andrade, C.K.Z.; Goulart, M.O.F.; Castro, S.L.; Pinto, A.V. Bioorg Med Chem 2010, 18, 3224-3230

3-Arylamino and 3-Alkoxy-nor-β-lapachone Derivatives: Synthesis and Cytotoxicity against Cancer Cell Lines

Júnior, E.N.S.; Deus, C.F.; Cavalcanti, B.C.; Pessoa, C.; Lotufo, L.V.C.; Montenegro, R.C.; Moraes, M.O.; Pinto, M.C.F.R.; Simone, C.A.; Ferreira, V.F.; Goulart, M.O.F.; Andrade, C.K.Z.; Pinto, A.V. J Med Chem 2010, 53, 504-508

Novel Supramolecular Palladium Catalyst for the Asymmetric Reduction of Imines in Aqueous Media

Silva, W.A.; Rodrigues, M.T.; Shankaraiah, N.; Ferreira, R.B.; Andrade, C.K.Z.; Pilli, R.A.; Santos, L.S. Org Lett 2009, 11, 3238-3241

Hooker’s ‘lapachol peroxide’ revisited

Júnior, E.N.S.; Pinto, M.C.F.R.; Moura, K.C.G.; Simone, C.A.; Nascimento, C.J.; Andrade, C.K.Z.; Pinto, A.V. Tetrahedron Lett 2009, 50, 1575-1577

Design and Synthesis of Cyclic RGD Pentapeptoids by Consecutive Ugi Reactions

Vercillo, O.E.; Andrade, C.K.Z.; Wessjohann, L.A. Org Lett 2008, 10, 205-208

Synthesis of new chiral ionic liquids based on (−)-menthol and (−)-borneol

Matos, R.A.F.; Andrade, C.K.Z. Tetrahedron Lett 2008, 49, 1652-1655

Synthesis and anti-Trypanosoma cruzi activity of derivatives from nor-lapachones and lapachones

Júnior, E.N.S.; Souza, M.C.B.V.; Fernandes, M.C.; Barreto, R.F.S.M.; Pinto, M.C.F.R.; Lopes, F.A.; Simone, C.A.; Andrade, C.K.Z.; Pinto, A.V.; Ferreira, V.F.; Castro, S.L. Bioorg Med Chem 2008, 16, 5030-5038

Enantioselective total synthesis of (S)-(−)-quinolactacin B

Shankaraiah, N.; Silva, W.A.; Andrade, C.K.Z.; Santos, L.S. Tetrahedron Lett 2008, 49, 4289-4291

3-(2,4-Dibromo­anilino)-2,2-dimethyl-2,3-dihydro­naphtho[1,2-b]furan-4,5-dione: a new substituted aryl­amino nor-[beta]-lapachone derivative

Silva, E.N.; Simone, C.A.; Goulart, M.O.F.; Andrade, C.K.Z.; Silva, R.S.F.; Pinto, A.V. Acta Crystaloogr E 2008, 64, o2348

Microwave assisted solvent-, support- and catalyst-free synthesis of enaminones

Andrade, C.K.Z. ARKIVOC 2008, 2008, 226-232

Computational Approach for the Design of AP1867 Analogs: Aiming at New Synthetic Routes for Potential Immunosuppressant Agents 

Andrade, C.K.Z.; Silva, W.A.; Maia, E.R. J Biomol Struct Dyn 2007, 25, 35-48

Organo-niobate Ionic Liquids: Synthesis, Characterization and Application as Acid Catalyst in Pechmann Reactions

Soares, V.C.D.; Alvez, M.B.; Souza, E.R.; Pinto, I.O.; Rubim, J.C.; Andrade, C.K.Z.; Suarez, P.A.Z. Int J Mol Sci 2007, 8, 392-398

One-Step Reduction of Chalcones to Saturated Alcohols by Ammonium Formate/Palladium on Carbon: A Versatile Method

Andrade, C.K.Z.; Silva, W.A. Lett Org Chem 2006, 3, 39-41 

3-(1,3-Benzodioxol-5-yl)-1-(4-methoxyphenyl)prop-2-enone

Andrade, C.K.Z.; Silva, W.A.; Vecanto, I.; Lariucci, C. Acta Crystallogr E 2006, 62, o1033-o1035

Revisiting the Passerini Reaction under Eco-Friendly Reaction Conditions

Andrade, C.K.Z.; Takada, S.C.S.; Suarez, P.A.Z.; Alvez, M.B. Synlett 2006, 2006, 1539-1542

Recent Applications of Niobium Catalysts in Organic Synthesis

Andrade, C.K.Z.; Rocha, R.O. Mini Rev Org Chem 2006, 3, 271-280

Environmentally Benign Solvents in Organic Synthesis: Current Topics

Andrade, C.K.Z.; Alves, L.M. Curr Org Chem 2005, 9, 195-218

Studies on the niobium pentachloride-mediated nucleophilic additions to an enantiopure cyclic N-acyliminium ion derived from (S)-malic acid

Andrade, C.K.Z.; Russowsky, D.; Rocha, R.O.; Godoy, M.N. J Braz Chem Soc 2005, 16, 535-539

Nucleophilic Additions of Niobium Enolates of Oxazolidinones to Aromatic Aldehydes and Aldimines

Andrade, C.K.Z.; Alves, L.M.; Kalil, P.P.; Rocha, R.O.; Panisset, C.M.A.; Lett Org Chem 2004, 1, 109-111

Intramolecular ene reactions catalyzed by NbCl5, TaCl5 and InCl3

Andrade, C.K.Z.; Vercillo, O.E.; Rodrigues, J.P.; Silveira, D.P. J Braz Chem Soc 2004, 15, 813-817

Niobium Pentachloride in Organic Synthesis: Applications and Perspectives

Andrade, C.K.Z. Curr Org Synth 2004, 1, 333- 353

Molecular Sieves in Ionic Liquids as an Efficient and Recyclable Medium for the Synthesis of Imines

Andrade, C.K.Z.; Suarez, P.A.Z.; Takada, S.C.; Alves, L.M.; Rodrigues, J.P.; Brandão, R.F.; Soares, V.C. Synlett 2004, 2004, 2135-2138

Niobium Pentachloride-mediated Nucleophilic Additions to Cyclic N-Acyliminium Ions

Andrade, C.K.Z.; Matos, R.A. Synlett 2003, 2003, 1189-1191

DCC/DMAP-Mediated Coupling of Carboxylic Acids with Oxazolidinones and Thiazolidinethiones

Andrade, C.K.Z.; Rocha, R.O.; Vercillo, O.E.; Silva, W.A.; Matos, R.A. Synlett 2003, 2003, 2351-2352

Allylation of aldimines promoted by NbCl5 

Andrade, C.K.Z.; Oliveira, G.R. Tetrahedron Lett 2002, 43, 1935-1937

NbCl5: A Novel Lewis Acid in Allylation Reactions

Andrade, C.K.Z.; Azevedo, N.R.; Oliveira, G.R. Synthesis 2002, 2002, 928-936

Niobium(V) chloride-mediated allylation of aldehydes. Scope and stereoselectivity 

Andrade, C.K.Z.; Azevedo, N.R. Tetrahedron Lett 2001, 42, 6473-6476